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Orion Pharma (Ireland) Ltd

Orion Pharma (Ireland) Ltd
c/o Allphar Services Ltd, 4045 Kingswood Road, Citywest Business Park, Co Dublin,
Telephone: +353 1 428 7777
Fax: +353 1 428 7776
Summary of Product Characteristics last updated on medicines.ie: 27/06/2011
SPC Entrydil S.R. 120mg Tablets

When a pharmaceutical company changes an SPC or PIL, a new version is published on medicines.ie. For each version, we show the dates it was published on medicines.ie and the reasons for change.

Updated on 27/06/2011 and displayed until Current
Reasons for adding or updating:
  • Correction of spelling/typing errors
Date of revision of text on the SPC:   01-Mar-2011
Legal Category:   Product subject to medical prescription which may be renewed (B)

Free-text change information supplied by the pharmaceutical company

Correction of errors in previous text
Updated on 21/03/2011 and displayed until 27/06/2011
Reasons for adding or updating:
  • Change to section 4.2 - Posology and method of administration
  • Change to section 4.3 - Contraindications
  • Change to section 4.4 - Special warnings and precautions for use
  • Change to section 4.5 - Interaction with other medicinal products and other forms of interaction
  • Change to section 4.6 - Pregnancy and lactation
  • Change to section 4.7 - Effects on ability to drive and use machines
  • Change to section 4.8 - Undesirable effects
  • Change to section 10 - Date of revision of the text
Date of revision of text on the SPC:   01-Mar-2011
Legal Category:   Product subject to medical prescription which may be renewed (B)

Free-text change information supplied by the pharmaceutical company

In section 4.2 the following text has been added:

Children (below 18 years of age):

 

There are no data available on use of diltiazem in children below the age of 18 years, and diltiazem is not recommended for use in children.

In section 4.3 the following text has been changed and added:

The 3rd bullet point has been changed to '......40 beats per minute'.

The 7th bullet point has added....'pulmonary congestion'

In section 4.4 the following text has been added: ....with impaired renal function or patients with renal or hepatic impairment

3. Prior to general anaesthesia, the anaesethist must be informed of ongoing diltiazem treatment. Depression of cardiac contractility, conductivity and automaticity, as well as the vascular dilatation associated with anaesthetics such as enflurane, halothane and isoflurane, may be potentiated by calcium channel blockers.

 

4. The risk of raised creatine kinease, myopathy and rhabdomyolisis due to statins (metabolised by CYP3A4) may be increased in case of a concomitant use of diltiazem. Closer monitoring for signs and symptoms is warranted in such case.

 

5. Calcium channel blocking agents, such as diltiazem, may be associated with mood   changes, including depression

 

6. Like other calcium channel antagonists, diltiazem has an inhibitory effect on intestinal motility. Therefore it should be used with caution in patients at risk to develop an intestinal obstruction.

In section 4.5, the following text has been added: In all the patients treated with calcium antagonists, the prescription of nitrate derivatives should only be carried out at gradually increasing doses.

-       .  The combination of diltiazem with an alpha-antagonist should be considered only with the strict monitoring of the blood pressure.

 

-      Dantrolene (infusion) a lethal ventricular fibrillation is regularly observed in animals when intravenous verapamil and dantrolene are administered concomitantly.  The combination of calcium antagonist and dantrolene is therefore potentially dangerous

       (see section 4.3 Contraindications).

 

Due to the potential for additive effects, caution and careful titration are necessary in patients receiving diltiazem concomitantly with other agents known to affect cardiac contractility and/or conduction.

In section 4.5, the following text has been added:

-       The patient should be carefully monitored when initiating or discontinuing rifampicin treatment.


-       Patients currently receiving diltiazem therapy should be carefully monitored when initiating or discontinuing therapy with anti-H2 agents. An adjustment in diltiazem daily dose may be necessary.

Under the subheading'Effect of diltiazem onother drugs, the following has been added:
4th paragraph-

-       Special care should be taken when prescribing short-acting benzodiazepines metabolized by the CYP3A4 pathway in patients using diltiazem.

In section 4.6 the following text has been added: There is very limited data from the use of diltiazem in pregnant patients.
....as well as in women of child-bearing potential not using effective contraception.

If use of diltiazem is considered medically essential, an alternative method of infant feeding should be instituted.


In section 4.7 the following text has been added: However, no studies have been performed.

In section 4.8 the foolowing information has been presented in a table format:

The following CIOMS frequency rating is used, when applicable: Very common (≥1/10); common (≥1/100 to <1/10); uncommon (≥1/1,000 to ≤1/100); rare (≥1/10,000 to ≤1/1,000); very rare (≤1/10,000); not known (cannot be estimated from the available data). Within each frequency grouping, adverse events are presented in order of decreasing seriousness

 

 

Very Common

Common

Uncommon

Rare

Not Known

Blood and

lymphatic system

disorders

 

 

 

 

Thrombocytopenia

Psychiatric

disorders

 

 

nervousness,

insomnia

 

Mood changes

(including

depression)

Nervous system

disorders

 

headache,

dizziness

 

 

extrapyramidal

syndrome

Cardiac

disorders

 

atrioventricular

block (may be

of first, second

or third degree;

bundle branch

block may

occur),

palpitations

bradycardia

 

Sinotrial block,

congestive heart

failure, syncope

Vascular

disorders

 

flushing

orthostatic

hypotension

 

Vasculitis

(including

leukocytoclastic

vasculitis)

Gastrointestinal

disorders

 

constipation,

dyspepsia,

gastric pain,

nausea

vomiting,

diarrhoea

dry mouth

Gingival

hyperplasia

Hepatobiliary

disorders

 

 

hepatic

enzymes

increase (AST,

ALT, LDH,

ALP increase)

 

Hepatitis

Musculoskeletal

and connective

tissue disorders

 

 

 

 

Arthralgia

Skin and

subcutaneous

tissue disorders

 

erythema

 

urticaria

Photosensitivity

(including

lichenoid keratosis

at sun exposed skin

areas),

angioneurotic

oedema, erythema

multiforme

(including Steven-

Johnson's syndrome and toxic epidermal

necrolysis),

sweating, exfoliative

dermatitis, acute

generalized

exanthematous

pustulosis,

occasionally

desquamative

erythema with or

without fever

Reproductive

system and

breast disorders

 

 

 

 

Gynecomastia

General

disorders and

administration

site conditions

lower limb

oedema (peripheral oedema)

malaise

 

 

Asthenia/fatigue

 

As with some other calcium channel blockers, exceptional cases of extrapyramidal symptoms and gynaecomastia have been reported, reversible after discontinuation of calcium antagonists. Raised creatine kinase, myopathy and rhabdomyolisis due to statins metabolised by the CYP3A4 system when taken concomitantly with diltiazem, see section 4.5, Interactions with Other Medicinal Products and Other Forms of Interaction.



In section 10 date of revision of text has been changed to March 2011

In section 4.7 the following text has been added: However, no studies have been performed.In section 4.8 the foolowing information has been presented in a table format:In section 10 date of revision of text has been changed to March 2011

In section 4.7 the following text has been added: However, no studies have been performed.In section 4.8 the foolowing information has been presented in a table format:In section 10 date of revision of text has been changed to March 2011

In section 4.7 the following text has been added: However, no studies have been performed.In section 4.8 the foolowing information has been presented in a table format:In section 10 date of revision of text has been changed to March 2011

In section 4.7 the following text has been added: However, no studies have been performed.In section 4.8 the foolowing information has been presented in a table format:In section 10 date of revision of text has been changed to March 2011

In section 4.7 the following text has been added: However, no studies have been performed.In section 4.8 the foolowing information has been presented in a table format:In section 10 date of revision of text has been changed to March 2011

In section 4.7 the following text has been added: However, no studies have been performed.In section 4.8 the foolowing information has been presented in a table format:In section 10 date of revision of text has been changed to March 2011
Updated on 13/07/2009 and displayed until 21/03/2011
Reasons for adding or updating:
  • Change to section 10 - Date of revision of the text
Date of revision of text on the SPC:   01-Jun-2009
Legal Category:   Product subject to medical prescription which may be renewed (B)

Free-text change information supplied by the pharmaceutical company

Section 10 (date of revision of text) has changed to June 2009
Updated on 18/08/2006 and displayed until 13/07/2009
Reasons for adding or updating:
  • Change to section 8 - MA number
  • Change to section 10 - Date of revision of the text
Date of revision of text on the SPC:   06/2006
Legal Category:   prescription only

Free-text change information supplied by the pharmaceutical company

Amended MA number and chane to partial revision of text

Updated on 24/11/2003 and displayed until 18/08/2006
Reasons for adding or updating:
  • New SPC for medicines.ie

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Active Ingredients

 
   Diltiazem Hydrochloride

Versions

 
27/06/2011 to Current
21/03/2011 to 27/06/2011
13/07/2009 to 21/03/2011
18/08/2006 to 13/07/2009
24/11/2003 to 18/08/2006
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Registered Address: Franklin House, 140 Pembroke Road, Dublin 4, Ireland
Registered Number: 254776
Tel: (353 1) 6603350 Fax: (353 1) 6686672 Email: info@ipha.ie

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