go to medicines.ie homepage
  • Home  |  
  • About  |  
  • Links  |  
  • Help
Font Size
Search for:  
select
select
  • SPCs and PILs
  • SPCs Only
  • PILs Only
  Advanced Search
  • What's
    New
      
  • Browse
    Medicines
      
  • Browse
    Active Ingredients
      
  • Browse
    Companies
      
  • Codes
    of Practice
      
  • Adverse
    Reaction Reporting


This is an X-PIL, which is a text only patient information leaflet, designed for people with sight problems.


Novo Nordisk Limited

Novo Nordisk Limited
3/4 Upper Pembroke Street, Dublin 2,
Telephone: +353 1 678 5989
Telephone: 1850 665 665
Fax: +353 1 676 3259
Medical Information e-mail: www.novonordisk.ie


Patient Information Leaflet last updated on medicines.ie: 16/12/2011
XPIL Trisequens

Table of Contents

  • PACKAGE LEAFLET: INFORMATION FOR THE USER
  • 1. What Trisequens® is and what it is used for
  • 2. Before you take Trisequens®
  • 3. How to take Trisequens®
  • 4. Possible side effects
  • 5. How To Store Trisequens®
  • 6. Further Information
  • USER INSTRUCTIONS

PACKAGE LEAFLET: INFORMATION FOR THE USER

Trisequens®

film-coated tablets

Estradiol and norethisterone acetate

Read this entire leaflet carefully before you start taking this medicine

  • Keep this leaflet. You may need to read it again.
  • If you have any further questions, ask your doctor or pharmacist.
  • This medicine has been prescribed for you. Do not pass it on to others. It may harm them, even if their symptoms are the same as yours.
  • If any of the side effects get serious, or if you notice any side effects not listed in this leaflet, please tell your doctor or pharmacist.

In this leaflet:

1. What Trisequens® is and what it is used for
2. Before you take Trisequens®
3. How to take Trisequens®
4. Possible side effects
5. How to store Trisequens®
6. Further information

Go to top of the page

1. What Trisequens® is and what it is used for

Trisequens® is a sequential combined Hormone Replacement Therapy (HRT) which is taken every day without interuption. It contains two types of female hormones, an oestrogen and a progestogen. Trisequens® is used in post-menopausal women with at least 6 months since their last natural period.

Trisequens® is used for:

Relief of symptoms occurring after menopause

During the menopause, the amount of the oestrogen produced by a woman’s body drops. This can cause symptoms such as hot face, neck and chest (“hot flushes”). Trisequens® alleviates these symptoms after menopause. You will only be prescribed Trisequens® if your symptoms seriously hinder your daily life.

Prevention of osteoporosis

After the menopause some women may develop fragile bones (osteoporosis). You should discuss all available options with your doctor. If you are at an increased risk of fractures due to osteoporosis and other medicines are not suitable for you, you can use Trisequens® to prevent osteoporosis after menopause.

The experience of treating women older than 65 years is limited.

Go to top of the page

2. Before you take Trisequens®

Medical history and regular check-ups

The use of HRT carries risks which need to be considered when deciding whether to start taking it, or whether to carry on taking it.

The experience in treating women with a premature menopause (due to ovarian failure or surgery) is limited. If you have a premature menopause the risks of using HRT may be different. Please talk to your doctor.

Before you start (or restart) HRT, your doctor will ask about your own and your family’s medical history. Your doctor may decide to perform a physical examination. This may include an examination of your breasts and/or an internal examination, if necessary.

Once you have started on Trisequens® you should see your doctor for regular check-ups (at least once a year). At these check-ups, discuss with your doctor the benefits and risks of continuing with Trisequens®.

Go for regular breast screening, as recommended by your doctor.

Do not take Trisequens®

If any of the following applies to you. If you are not sure about any of the points below, talk to your doctor before taking Trisequens®,

Do not take Trisequens®

  • If you have or have ever had breast cancer, or if you are suspected of having it
  • If you have cancer which is sensitive to oestrogens, such as cancer of the womb lining (endometrium), or if you are suspected of having it
  • If you have any unexplained vaginal bleeding
  • If you have excessive thickening of the womb lining (endometrial hyperplasia) that is not being treated.
  • If you have or have ever had a blood clot in a vein (thrombosis), such as in the legs (deep venous thrombosis) or the lungs (pulmonary embolism)
  • If you have a blood clotting disorder (such as protein C, protein S, or antithrombin deficiency)
  • If you have or recently have had a disease caused by blood clots in the arteries, such as a heart attack, stroke or angina
  • If you have or have ever had a liver disease and your liver function tests have not returned to normal
  • If you have a rare blood problem called “porphyria” which is passed down in families (inherited)
  • If you are allergic (hypersensitive) to estradiol, norethisterone acetate or any of the other ingredients of Trisequens® (listed in section 6 Further information)

If any of the above conditions appear for the first time while taking Trisequens®, stop taking it at once and consult your doctor immediately.

When to take special care with Trisequens®

Tell your doctor if you have ever had any of the following problems, before you start the treatment, as these may return or become worse during treatment with Trisequens®. If so, you should see your doctor more often for check-ups:

  • fibroids inside your womb
  • growth of womb lining outside your womb (endometriosis) or a history of excessive growth of the womb lining (endometrial hyperplasia)
  • increased risk of developing blood clots (see “Blood clots in a vein (thrombosis)”)
  • increased risk of getting a oestrogen-sensitive cancer (such as having a mother, sister or grandmother who has had breast cancer)
  • high blood pressure.
  • a liver disorder, such as a benign liver tumour
  • diabetes
  • gallstones
  • migraine or severe headaches.
  • a disease of the immune system that affects many organs of the body (systemic lupus erythematosus, SLE)
  • epilepsy
  • asthma
  • a disease affecting the eardrum and hearing (otosclerosis)
  • a very high level of fat in your blood (triglycerides)
  • fluid retention due to cardiac or kidney problems

Stop taking Trisequens® and see a doctor immediately

If you notice any of the following when taking HRT:

  • any of the conditions mentioned in the ‘DO NOT take Trisequens®’ section
  • yellowing of your skin or the whites of your eyes (jaundice). These may be signs of a liver disease
  • a large rise in your blood pressure (symptoms may be headache, tiredness, dizziness).
  • migraine-like headaches which happen for the first time.
  • if you become pregnant
  • if you notice signs of a blood clot, such as:
    • painful swelling and redness of the legs
    • sudden chest pain
    • difficulty in breathing

For more information, see ‘Blood clots in a vein (thrombosis)’

Note: Trisequens® is not a contraceptive. If it is less than 12 months since your last menstrual period or you are under 50 years old, you may still need to use additional contraception to prevent pregnancy. Speak to your doctor for advice.

HRT and cancer

Excessive thickening of the lining of the womb (endometrial hyperplasia) and cancer of the lining of the womb (endometrial cancer)

Taking oestrogen-only HRT will increase the risk of excessive thickening of the lining of the womb (endometrial hyperplasia) and cancer of the womb lining (endometrial cancer).

The progestogen in Trisequens® protects you from this extra risk.

Unexpected bleeding

You will have a bleed once a month (so-called withdrawal bleed) while taking Trisequens®. But, if you have unexpected bleeding or drops of blood (spotting) besides your monthly bleeding, which:

  • carries on for more than the first 6 months
  • starts after you have been taking Trisequens® more than 6 months
  • carries on after you have stopped taking Trisequens®

see your doctor as soon as possible

Breast cancer

Evidence suggests that taking combined oestrogen-progestogen and possibly also oestrogen-only HRT increases the risk of breast cancer. The extra risk depends on how long you take HRT. The additional risk becomes clear within a few years. However, it returns to normal within a few years (at most 5) after stopping treatment.

Compare

Women aged 50 to 79 who are not taking HRT, on average, 9 to 14 in 1000 will be diagnosed with breast cancer over a 5-year period. For women aged 50 to 79 who are taking oestrogen-progestogen HRT over 5 years, there will be 13 to 20 cases in 1000 users (i.e. an extra 4 to 6 cases).

  • Regularly check your breasts. See your doctor if you notice any changes such as:
    • dimpling of the skin
    • changes in the nipple
    • any lumps you can see or feel

Ovarian cancer

Ovarian cancer is rare. A slightly increased risk of ovarian cancer has been reported in women taking HRT for at least 5 to 10 years.

Compare

Women aged 50 to 69 who are not taking HRT, on average about 2 women in 1000 will be diagnosed with ovarian cancer over a 5-year period. For women who have been taking HRT for 5 years, there will be between 2 and 3 cases per 1000 users (i.e. up to 1 extra case).

Effect of HRT on heart and circulation

Blood clots in a vein (thrombosis)

The risk of blood clots in the veins is about 1.3 to 3- times higher in HRT users than in non-users, especially during the first year of taking it.

Blood clots can be serious, and if one travels to the lungs, it can cause chest pain, breathlessness, fainting or even death.

You are more likely to get a blood clot in your veins as you get older and if any of the following applies to you. Inform your doctor if any of these situations applies to you:

  • you are unable to walk for a long time because of major surgery, injury or illness (see also section 3, If you need to have surgery)
  • you are seriously overweight (BMI >30 kg/m2)
  • you have any blood clotting problem that needs long-term treatment with a medicine used to prevent blood clots
  • if any of your close relatives has ever had a blood clot in the leg, lung or an other organ
  • you have systemic lupus erythematosus (SLE)
  • you have cancer.

For signs of a blood clot, see “Stop taking Trisequens® and see a doctor immediately”.

Compare

Looking at women in their 50s who are not taking HRT, on average, over a 5-year period, 4 to 7 in 1000 would be expected to get a blood clot in a vein.

For women in their 50s who have been taking oestrogen-progestogen HRT for over 5 years, there will be 9 to 12 cases in 1000 users (i.e. an extra 5 cases).

Heart disease (heart attack)

There is no evidence that HRT will prevent a heart attack.

Women over the age of 60 years who use oestrogen-progestogen HRT are slightly more likely to develop heart disease than those not taking any HRT.

Stroke

The risk of getting stroke is about 1.5 times higher in HRT users than in non-users. The number of extra cases of stroke due to use of HRT will increase with age.

Compare

Looking at women in their 50s who are not taking HRT, on average, 8 in 1000 would be expected to have a stroke over a 5-year period. For women in their 50s who are taking HRT, there will be 11 cases in 1000 users, over 5 years (i.e. an extra 3 cases).

Other conditions

  • HRT will not prevent memory loss. There is some evidence of a higher risk of memory loss in women who start using HRT after the age of 65. Speak to your doctor for advice.

Using other medicines

Some medicines may interfere with the effect of Trisequens®. This might lead to irregular bleeding. This applies to the following medicines:

  • Medicines for epilepsy (such as phenobarbital, phenytoin and carbamazepin)
  • Medicines for tuberculosis (such as rifampicin, rifabutin)
  • Medicines for HIV infection (such as nevirapine, efavirenz, ritonavir and nelfinavir)
  • Herbal remedies containing St John’s Wort (Hypericum perforatum).

Other medicines may increase the effects of Trisequens®:

  • Drugs containing ketoconazole (a fungicide)

Concomitant administration of cyclosporine may cause increased blood levels of cyclosporine.

Please tell your doctor or pharmacist if you are taking or have recently taken any other medicines including medicines obtained without a prescription, herbal medicines or other natural products.

Taking Trisequens® with food and drink

The tablets can be taken with or without food and drink.

Laboratory tests

If you need a blood test, tell your doctor or the laboratory staff that you are taking Trisequens®, because this medicine can affect the results of some tests.

Pregnancy and breast-feeding

Trisequens® is for use in post-menopausal women only. If you become pregnant, stop taking Trisequens® and contact your doctor. You should not use Trisequens® if you are breast-feeding.

Driving and using machines

Trisequens® has no known effect on the ability to drive or use machines.

Important information about some of the ingredients in Trisequens®

Trisequens® contains lactose monohydrate. If you have been told by your doctor that you have an intolerance to some sugars, contact your doctor before taking Trisequens®.

Go to top of the page

3. How to take Trisequens®

Always take Trisequens® exactly as your doctor has told you. You should check with your doctor or pharmacist if you are unsure.

If you are not switching from another hormone replacement therapy you can start treatment with Trisequens® on any convenient day. If you are switching from another hormone replacement therapy ask your doctor when you should start treatment with Trisequens®.

Take one tablet once a day, at about the same time each day.

Each pack contains 28 tablets

Days 1 - 12 Take one blue tablet everyday for 12 days

Days 13 - 22 Take one white tablet everyday for 10 days

Days 23 - 28 Take one red tablet everyday for 6 days

Take the tablets with a glass of water.

Once you have finished the pack, start a new pack continuing the treatment without interruption. A menstruation-like bleeding usually occurs at the beginning of a new pack.

For further information on the use of the calendar pack, see USER INSTRUCTIONS at the end of the package leaflet.

Your doctor will aim to prescribe the lowest dose to treat your symptom for as short as necessary. Speak to your doctor if you think this dose is too strong or not strong enough. Talk to your doctor if you do not experience symptom relief after 3 months of treatment. You should only continue treatment as long as the benefit outweighs the risk.

If you take more Trisequens® than you should

If you have taken more Trisequens® tablets than you should, talk to a doctor or pharmacist.

An overdose of Trisequens® could make you feel sick or vomit.

If you forget to take Trisequens®

Do not take a double dose to make up for a forgotten individual dose. If you forget to take your tablet at the usual time, take it within the next 12 hours. If more than 12 hours have gone by, start again as normal the next day. Do not take a double dose to make up for a forgotten tablet.

Forgetting a dose may increase the likelihood of breakthrough bleeding and spotting.

If you stop taking Trisequens®

If you would like to stop your treatment with Trisequens® for any reason, please discuss your decision with your doctor, who will explain the effects of stopping treatment and discuss other possibilities with you. If you have any further questions on the use of this product, ask your doctor or pharmacist.

If you need to have surgery

If you are going to have surgery, tell the surgeon that you are taking Trisequens®. You may need to stop taking Trisequens® about 4 to 6 weeks before the operation to reduce the risk of a blood clot (see section 2, Blood clots in a vein). Ask your doctor when you can start taking Trisequens® again.

Go to top of the page

4. Possible side effects

The following diseases are reported more often in women using HRT compared to women not using HRT:

  • breast cancer
  • abnormal growth or cancer of the lining of the womb (endometrial hyperplasia or cancer)
  • ovarian cancer
  • blood clots in the veins of the legs or lungs (venous thromboembolism)
  • heart disease
  • stroke
  • probable memory loss if HRT is started over the age of 65

For more information about these side effects, see Section 2.

Hypersensitivity/allergy

(uncommon side effects - Affects 1 in 10 users in 1,000)

Though it is an uncommon event, hypersensitivity/allergy may occur. Signs of hypersensitivity/allergy may include one or more of the following symptoms: hives, itching, swelling, difficulty in breathing, low blood pressure (paleness and coldness of skin, rapid heart beat), feeling dizzy, sweating, which could be signs of anaphylactic reaction/shock. If one of the mentioned symptoms appears, stop taking Trisequens® and seek immediate medical help.

The frequency of possible side effects listed below is defined using the following convention:

Very common (affects more than 1 user in 10)

Common (affects 1 to 10 users in 100)

Uncommon (affects 1 to 10 users in 1,000)

Rare (affects 1 to 10 users in 10,000)

Very rare (affects less than 1 user in 10,000)

Not known (frequency cannot be estimated from the available data)

Very common side effects

  • Breast pain or breast tenderness
  • Irregular periods or excessive bleeding during your periods

Common side effects

  • Headache
  • Weight gain caused by fluid retention
  • Vaginal inflammation
  • Vaginal infection with a fungus
  • Migraine, new or worse than before
  • Depression, new or worse than before
  • Nausea
  • Abdominal pain, swelling or discomfort
  • Enlargement or swelling of the breasts (breast oedema)
  • Back pain
  • Leg cramps
  • Uterine fibroid (benign tumour), aggravation, occurrence or reoccurrence
  • Swelling of arms and legs (peripheral oedema)
  • Weight increase

Uncommon side effects

  • Bloating or flatulence
  • Acne
  • Hair loss (alopecia)
  • Abnormal (male pattern) hair growth
  • Itching or hives (urticaria)
  • Inflammation of a vein (superficial thrombophlebitis)
  • Drug ineffective
  • Allergic reaction
  • Endometrial hyperplasia (excessive growth of the lining of the womb)
  • Painful periods
  • Nervousness

Rare side effects

  • Pulmonary embolism (blood clot) (See also Blood clots in section 2 Before you take Trisequens®)
  • Deep inflammation of a vein associated with thrombosis (blood clot)

Very rare side effects

  • Cancer of the lining of the womb (endometrial cancer)
  • Increase in blood pressure or worsening of high blood pressure
  • Gallbladder disease, gallstones occurrence/reoccurrence or aggravated
  • Excessive secretion of sebum, skin eruption
  • Acute or recurring attack of oedema (angioneurotic oedema)
  • Insomnia, dizziness, anxiety
  • Change in sexual desire
  • Visual disturbances
  • Weight decreased
  • Vomiting
  • Heartburn
  • Vaginal and genital itching
  • Heart attack and stroke

If any of the side effects get serious, or if you notice any side effects not listed in this leaflet, please tell your doctor or pharmacist.

The following side effects have been reported with other HRTs:

  • various skin disorders:
    • discoloration of the skin especially of the face or neck known as “pregnancy patches” (chloasma)
    • painful reddish skin nodules (erythema nodosum)
    • rash with target-shaped reddening or sores (erythema multiforme)
Go to top of the page

5. How To Store Trisequens®

Keep out of the reach and sight of children.

Do not use Trisequens® after the expiry date which is stated on the label and outer carton after ‘EXP’.

The expiry date refers to the last day of that month.

Store below 25°C. Do not refrigerate.

Keep the container in the outer carton in order to protect from light.

Medicines should not be disposed of via wastewater or household waste. Ask your pharmacist how to dispose of medicines no longer required. These measures will help to protect the environment.

Go to top of the page

6. Further Information

What Trisequens® contains

  • The active substances are estradiol and norethisterone acetate.
  • The blue film-coated tablet contains: estradiol 2 mg (as estradiol hemihydrate).
  • The white film-coated tablet contains: estradiol 2 mg (as estradiol hemihydrate) and norethisterone acetate 1 mg.
  • The red film-coated tablet contains: estradiol 1 mg (as estradiol hemihydrate).
  • The other ingredients are: lactose monohydrate, maize starch, hydroxypropylcellulose, talc and magnesium stearate.
  • Film-coating (blue tablets) contain: hypromellose, talc, titanium dioxide (E171), indigo carmine (E132) and macrogol 400.
  • Film-coating (white tablets) contain: hypromellose, triacetin and talc.
  • Film-coating (red tablets) contain: hypromellose, talc, titanium dioxide (E171), red iron oxide (E172) and propylene glycol.

What Trisequens® looks like and contents of the pack

The film-coated tablets are round with a diameter of 6 mm. The blue tablets are engraved with NOVO 280. The white tablets are engraved with NOVO 281. The red tablets are engraved with NOVO 282.

Each pack of 28 tablets contains 12 blue tablets, 10 white tablets and 6 red tablets.

Pack sizes available:

  • 1×28 film-coated tablets

Marketing Authorisation Holder and Manufacturer:

Novo Nordisk A/S
Novo Allé
DK-2880 Bagsværd
Denmark

Further information on Trisequens® is available to the medical and allied professions from:

Novo Nordisk Limited
3-4 Upper Pembroke Street
Dublin 2
Phone (01) 6785989
Fax (01) 6763259
Go to top of the page

This leaflet was last approved in: 12/2011

USER INSTRUCTIONS

How to use the calendar pack

1. Set the day reminder

Turn the inner disc to set the day of the week opposite the little plastic tab.

2. Take the first day’s tablet

Break the plastic tab and tip out the first tablet.

3. Move the dial every day

On the next day simply move the transparent dial clockwise 1 space as indicated by the arrow. Tip out the next tablet. Remember to take only 1 tablet once a day.

You can only turn the transparent dial after the tablet in the opening has been removed.

Go to top of the page

Trisequens® is a trademark owned by Novo Nordisk FemCare AG, Switzerland

© 2011

Novo Nordisk A/S

8-2801-11-042-5



Link to this document from your website:
http://www.medicines.ie/medicine/14529/XPIL/Trisequens/

Document Links

 
  Link to this page
  View all medicines
from this company
View original PDF PIL
View document history
Bookmark and Share

Legal Categories

 
   Product subject to medical
prescription which may not
be renewed (A)
   Product subject to medical
prescription which may
be renewed (B)
   Product subject to
restricted prescription
(C)
   Supply through
general sale
   Supply through
pharmacy only

Active Ingredients

 
   Estradiol Hemihydrate
   Norethisterone acetate

  • Terms & Conditions | 
  • Accessibility | 
  • Privacy Statement | 
  • Contact Us

Registered Address: Franklin House, 140 Pembroke Road, Dublin 4, Ireland
Registered Number: 254776
Tel: (353 1) 6603350 Fax: (353 1) 6686672 Email: info@ipha.ie

This website is certified by Health On the Net Foundation. Click to verify.

This site complies with the HONcode standard for trustworthy health information: verify here.

logo